Keap1-Nrf2-IN-12 is a potentKeap1-Nrf2inhibitor with anIC₅₀value of 2.30 μM. Keap1-Nrf2-IN-12 shows metabolic stability in human liver microsomes^[1].

IC₅₀: 2.30 μM (Keap1-Nrf2)^[1].

Keap1-Nrf2-IN-12 (compound 9a) shows metabolic stability in human liver microsomes with slight changes (97.7% remained) after 90 min of incubation^[1].

592.64

C₂₆H₂₈N₂O₁₀S₂

2250082-04-1

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.