| CAS NO: | 261766-73-8 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 25mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| 200mg | 电议 |
| 生物活性 | 5-HT4 antagonist 1 is a5-HT4receptorantagonist with apKiof 9.6. | ||||||||||||
| IC50& Target |
| ||||||||||||
| 体外研究 (In Vitro) | 5-HT4 antagonist 1 (compound 6b) is a 5-HT4receptor antagonist with a pKiof 9.6. | ||||||||||||
| 体内研究 (In Vivo) | 5-HT4 antagonist 1 (compound 6b) demonstrates good exposure and prolongs t1/2in other species, including the mouse (t1/27 h), rat (t1/212 h) and mini-pig (t1/221 h). In Phase I clinical trial, it is found that 5-HT4 antagonist 1 has good oral bioavailability with a steady state plasma t1/2of >100 h[1]. | ||||||||||||
| 分子量 | 480.62 | ||||||||||||
| 性状 | Solid | ||||||||||||
| Formula | C23H36N4O5S | ||||||||||||
| CAS 号 | 261766-73-8 | ||||||||||||
| 运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| 储存方式 |
|
m.cnreagent.com