EZH2-IN-5

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EZH2-IN-5

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

1403258-69-4

包装与价格：

产品介绍

EZH2-IN-5 是一种有效的EZH2抑制剂，对野生型和突变型 Tyr641 EZH2 的IC₅₀值分别为 1.52 nM 和 4.07 nM。

生物活性

EZH2-IN-5 is a potentEZH2inhibitor withIC₅₀values of 1.52 nM and 4.07 nM for wild-type and mutant Tyr641EZH2, respectively^[1].

IC₅₀& Target^[1]

EZH2 WT

1.52 nM (IC₅₀)

EZH2 Y641F mutant type

4.07 nM (IC₅₀)

体外研究
(In Vitro)

EZH2-IN-5 (compound 276) inhibits cell growth of WSUDLCL2 cell lines with an IC₅₀of 187.28 nM^[1].

分子量

517.50

Formula

C₂₆H₃₇BrN₄O₂

CAS 号

1403258-69-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.