UNC2399

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UNC2399

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:	2412791-72-9
包装:	1mg

产品介绍

UNC2399，一种生物素化的 UNC1999，是选择性的EZH2降解剂，对 EZH2 具有很高的体外效力，IC₅₀值为 17 nM。

生物活性

UNC2399, a biotinylated UNC1999, is a selectiveEZH2degrader, maintaining high in vitro potency forEZH2, with anIC₅₀of 17 nM^[1]^[2].

IC₅₀& Target^[1]

EZH2

17 nM (IC₅₀)

体外研究
(In Vitro)

UNC2399 (1-1000 nM) displays high in vitro potency (IC₅₀=17±2 nM) in the EZH2 radioactive biochemical assay^[1].
UNC2399 (100 μM) enriches EZH2 from HEK293T cell lysates^[1].

分子量

927.17

Formula

C₄₈H₆₆N₁₀O₇S

CAS 号

2412791-72-9

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.