CSV0C018875

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CSV0C018875

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

442150-41-6

包装与价格：

产品介绍

CSV0C018875 是一种基于喹啉的EHMT2/G9a抑制剂。 CSV0C018875 的细胞毒性低于 BIX-01294。

生物活性

CSV0C018875 is a quinoline-basedEHMT2/G9ainhibitor. CSV0C018875 exhibits lesser cytotoxicity than BIX-01294^[1].

IC₅₀& Target^[1]

G9a

体外研究
(In Vitro)

CSV0C018875 (2.5-20 μM; 48 hours) inhibits the levels of H3K9me2 modifications in the histones^[1].

Western Blot Analysis^[1]

Cell Line:	HEK293 cells
Concentration:	2.5 μM, 10 μM, 20 μM
Incubation Time:	48 hours
Result:	Inhibited the enzymatic activity of G9a in a dose-dependent manner in HEK293 cells.

分子量

312.79

Formula

C₁₈H₁₇ClN₂O

CAS 号

442150-41-6

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.