MA 2029 是一种选择性、口服活性和竞争性胃动素受体拮抗剂 (IC50\u003d4.9 nM)。
| Cas No. | 287206-61-5 |
| 化学名 | (S,Z)-N-((S,Z)-3-(3-(tert-butyl)-4-hydroxyphenyl)-1-(ethylimino)-1-hydroxypropan-2-yl)-2-((S)-3-(4-fluorophenyl)-N-methyl-2-(methylamino)propanamido)-3-methylbutanimidic acid |
| Canonical SMILES | CC/N=C(O)/[C@](/N=C(O)/[C@](N(C([C@](NC)([H])CC1=CC=C(F)C=C1)=O)C)([H])C(C)C)([H])CC2=CC(C(C)(C)C)=C(O)C=C2 |
| 分子式 | C31H45FN4O4 |
| 分子量 | 556.71 |
| 溶解度 | <11.13mg/ml in 1eq. HCl;<55.67mg/ml in DMSO |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |