PF-02575799

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PF-02575799

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

863491-70-7

包装与价格：

产品介绍

MTP-IN-1是微粒体甘油三酯转移蛋白 (microsomal triglyceride transfer protein (MTP)) 抑制剂，IC₅₀值为0.77±0.29 nM。

生物活性	PF-02575799 is amicrosomal triglyceride transfer protein (MTP)inhibitor with anIC₅₀of 0.77±0.29 nM.
IC₅₀& Target	IC50: 0.77±0.29 nM (MTP)^[1]
体外研究 (In Vitro)	PF-02575799 is compound 13 from the reference^[1].
体内研究 (In Vivo)	PF-02575799 produces appreciable triglyceride effects at its minimally effective dose (10 mg/kg). PF-02575799 significant increase alanine transaminase at 100 mg/kg^[1].
分子量	680.77
Formula	C₄₂H₃₇FN₄O₄
CAS 号	863491-70-7
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.