CALP1 TFA is acalmodulin(CaM)agonist (K_dof 88 μM) with binding to theCaMEF-hand/Ca²⁺-binding site. CALP1 TFA blocks calcium influx andapoptosis(IC₅₀of 44.78 μM) through inhibition ofcalcium channelopening. CALP1 TFA blocksglutamate receptor channelsand blocks a store-operated nonselective cation channel. CALP1 TFA activatesCaM-dependentphosphodiesteraseactivity^[1][2][3][4].

Kd: 88 μM (Calmodulin)^[4]

956.10

Solid

C₄₂H₇₆F₃N₉O₁₂

Val-Ala-Ile-Thr-Val-Leu-Val-Lys

VAITVLVK

Room temperature in continental US; may vary elsewhere.

Sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

H₂O : 16.67 mg/mL(17.44 mM;Need ultrasonic)

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80℃, 6 months; -20℃, 1 month (sealed storage, away from moisture)。-80℃ 储存时，请在 6 个月内使用，-20℃ 储存时，请在 1 个月内使用。