CCG-271423

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CCG-271423

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

2750413-88-6

包装与价格：

产品介绍

CCG-271423 是一种有效的选择性GRK5抑制剂，GRK5 和 GRK2 的IC₅₀值分别为 0.0021 μM 和 44 μM。CCG-271423 抑制心肌细胞收缩能力，降低 Ca²⁺瞬态。

生物活性	CCG-271423 is a potent and selectiveGRK5inhibitor withIC₅₀values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca²⁺transience^[1].
IC₅₀& Target	IC50: 0.0021 μM (GRK5) and 44 μM (GRK5)^[1]
体外研究 (In Vitro)	CCG-271423 (1 μM) does not alter cardiomyocyte contractility and decreases in Ca²⁺transience^[1].
分子量	466.53
Formula	C₂₈H₂₆N₄O₃
CAS 号	2750413-88-6
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.