| CAS NO: | 1052147-86-0 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 25mg | 电议 |
| CAS: | 1052147-86-0 |
| 分子式: | C30H34N4O |
| 分子量: | 466.62 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months; -20℃ 1 month |
| 研究领域: | Neurological Disease |
| Target: | Ki:0.58 nM (5-HT7 receptor), 188 nM (5-HT1A receptor), 142 nM (D2 receptor)[1] |
| 描述: | LP-211 is a selective and blood–brain barrier penetrant 5-HT7 receptor agonist, with a Ki of 0.58 nM, with high selectivity over 5-HT1A receptor (Ki, 188 nM) and D2 receptor (Ki, 142 nM). |
