| CAS NO: | 1300031-52-0 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| CAS: | 1300031-52-0 |
| 分子式: | C25H23ClN2O3 |
| 分子量: | 434.91 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | 22 nM (BRD4), 31 nM (BRD3), 41 nM (BRD2)[1] |
| 描述: | GSK1324726A is a potent, and selective inhibitor of BET proteins with high affinity to BRD2 (IC50=41 nM), BRD3 (IC50=31 nM), and BRD4(IC50=22 nM). |
