Palbociclib(PD 0332991)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
包装与价格:
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| 500mg | 电议 |
产品介绍
| 产品名称: | 帕布昔利布 |
| CAS: | 571190-30-2 |
| 分子式: | C24H29N7O2 |
| 分子量: | 447.53 |
| 纯度: | >98% |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | IC50: 9 nM (Cdk4/cyclin D3), 11 nM (Cdk4/cyclin D1), 16 nM (Cdk6/cyclin D2), 2000 nM (DYRK1A)[1] |
| 描述: | Palbociclib (PD 0332991) is a selective CDK4 and CDK6 inhibitor with IC50s of 11 and 16 nM, respectively. Palbociclib is a drug for the treatment of ER-positive and HER2-negative breast cancer. |