| CAS NO: | 755037-03-7 |
| 包装 | 价格(元) |
| 10mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| 产品名称: | 瑞格非尼 |
| CAS: | 755037-03-7 |
| 分子式: | C21H15ClF4N4O3 |
| 分子量: | 482.82 |
| 纯度: | ≥98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | IC50: 13 nM (VEGFR1), 4.2 nM (VEGFR2), 46 nM (VEGFR3), 22 nM (PDGFRβ), 7 nM (Kit), 1.5 nM (RET), 2.5 nM (Raf-1) |
| 描述: | Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM, 4.2 nM, 46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively. |
