| CAS NO: | 1942919-79-0 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| CAS: | 1942919-79-0 |
| 分子式: | C27H30Cl2F2N6O |
| 分子量: | 563.47 |
| 纯度: | ≥98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | IC50: 0.48 nM (JAK2 JH1), 31.63 nM (JAK1 JH1), 18.68 nM (JAK3 JH1), 10.76 nM (TYK2 JH1), 0.56 nM (FL JAK2 V617F), 0.58 nM (FL JAK2 wt)[1] |
| 描述: | NVP-BSK805 dihydrochloride is an ATP-competitive JAK2 inhibitor, with IC50 of 0.48 nM, 31.63 nM, 18.68 nM, and 10.76 nM for JAK2 JH1 (JAK homology 1), JAK1 JH1, JAK3 JH1, and TYK2 JH1, respectively. |
