| CAS NO: | 537049-40-4 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| CAS: | 537049-40-4 |
| 分子式: | C41H43N3O7S |
| 分子量: | 721.86 |
| 纯度: | ≥98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer/Infection |
| Target: | IC50: 4 nM (HDAC6), 1.27 μM (HDAC3), 1.27 μM (HDAC8), 1.40 μM (HDAC1), 3.35 μM (HDAC5), 3.71 μM (HDAC10), 3.79 μM (HDAC11), 4.31 μM (HDAC9), 6.27 μM (HDAC2), 9.7 μM (HDAC7), 17.3 μM (HDAC4)[1] |
| 描述: | Tubacin is a potent and selective inhibitor of HDAC6, with an IC50 value of 4 nM and approximately 350-fold selectivity over HDAC1. |
