| CAS NO: | 2341740-84-7 |
| 包装: | 5mg |
| 市场价: | 11560元 |
| CAS: | 2341740-84-7 |
| 分子式: | C44H42F3N7O12 |
| 分子量: | 917.84 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | PTK2/FAK:18 nM (IC50);Cereblon |
| 描述: | BI-3663 is a highly selective PTK2/FAK PROTAC, with cereblon ligands to hijack E3 ligases for PTK2 degradation. BI-3663 inhibits PTK2 with an IC50 of 18 nM. |
