| CAS NO: | 1645286-75-4 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| CAS: | 1645286-75-4 |
| 分子式: | C25H28N6O |
| 分子量: | 428.53 |
| 纯度: | ≥98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | IC50: 3 nM (TNKS1), 1 nM (TNKS2), 2.0 μM (PARP1), 0.5 μM (PARP2), >3 μM (PARP6)[1] |
| 描述: | AZ6102 is a potent dual TNKS1 and TNKS2 inhibitor, with IC50 of 3 nM and 1 nM, respectively, and alao has 100-fold selectivity against other PARP family enzymes, with IC50 of 2.0 μM, 0.5 μM, and >3 μM |
