| CAS NO: | 451492-95-8 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
| 50mg | 电议 |
| 100mg | 电议 |
| CAS: | 451492-95-8 |
| 分子式: | C27H28ClFN6O |
| 分子量: | 507.00 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | EGFR0.75 nM (IC50);ErbB219 nM (IC50);EGFRL858R0.51 nM (IC50);EGFRL858R/T790M2.3 nM (IC50);EGFRT790M0.79 nM (IC50) |
| 描述: | AV-412 free base (MP-412 free base) is an EGFR inhibitor with IC50s of 0.75, 0.5, 0.79, 2.3, 19 nM for EGFR, EGFRL858R, EGFRT790M, EGFRL858R/T790M and ErbB2, respectively. |
