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Oliceridine Racemate
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Oliceridine Racemate图片
CAS NO:1401028-25-8
包装与价格：
包装价格(元)
2mg电议
5mg电议
10mg电议
50mg电议
100mg电议
200mg电议

产品介绍
Oliceridine Racemate (TRV130 Racemate) 是 TRV130 的外消旋体。Oliceridine 是新颖的 MOR 激动剂，能够优先激活 G-protein 信号通路，而对 β-arrestin 的作用稍弱。
Cas No.1401028-25-8
Canonical SMILESCOC1=C(CNCCC(C2)(C3=NC=CC=C3)CCOC42CCCC4)SC=C1
分子式C22H30N2O2S
分子量386.55
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Oliceridine Racemate (TRV130 Racemate) is the racemate of Oliceridine. Oliceridine is a novel mu opioid receptor (MOR) agonist that preferentially activates G-protein versus β-arrestin signaling pathways coupled to MORs.

[1]. Altarifi AA, et al. Effects of acute and repeated treatment with the biased mu opioid receptor agonist TRV130 (oliceridine) on measures of antinociception, gastrointestinal function, and abuse liability in rodents. J Psychopharmacol. 2017 Jan 1:2698811166