EPZ-719 是一种新型有效的 SETD2 抑制剂（IC50 = 0.005 μM），与其他组蛋白甲基转移酶相比具有高选择性。
货号:ajcx37430
CAS:2697176-16-0
分子式:C22H31FN4O3S
分子量：450.57
溶解度:N/A
纯度：98%
存储：Store at -20°C
库存：现货

Background:

EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0.005 μM) with a high selectivity over other histone methyltransferases.

[1]. Lampe JW, et al. Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies. ACS Med Chem Lett. 2021 Aug 24;12(10):1539-1545.