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Bliretrigine
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Bliretrigine图片
规格:98%
分子量:352.43
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议

产品介绍
Bliretrigine 是一种钠通道 (sodium channel) 阻滞剂。Bliretrigine 有缓解疼痛的作用。
货号:ajcx38042
CAS:1233229-75-8
分子式:C20H24N4O2
分子量:352.43
溶解度:DMSO : 50 mg/mL (141.87 mM; Need ultrasonic)
纯度:98%
存储:Store at -20°C
库存:现货

Background:

Bliretrigine is a sodium channel blocker. Bliretrigine has the effect of relieving pain[1][2][3].

[1]. WHO Drug Information, Vol. 35, No. 4, 2021. Geneva: World Health Organization; 2022.
[2]. Yoshihiro OYAMADA, et al. External medicinal preparation containing N2-{[1-ethyl-6-(4-methylphenoxy)-1H-benzimidazol-2-yl]methyl}-L-alanineamide for treating and/or preventing peripheral neuropathic pain. Patent AU2019306705.
[3]. Hironori Kinoshita, et al. Preparation of N2-[(benzimidazol-2-yl or imidazo[4,5-b]pyridin-2-yl)methyl]amino acid amide derivatives as inhibitors of sensory neuron specific sodium channel (SNS). Patent AU2009331179.