Oleoyl-D-lysine is an inhibitor of glycine transporter 2a (GlyT2a).
货号:ajcx18798
CAS:N/A
分子式:C24H46N2O3•Na
分子量：433.6
溶解度:DMF: 10mg/mL,DMSO: 30mg/mL,Ethanol: 50mg/mL,PBS (pH 7.2): 0.25mg/mL
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Oleoyl-D-lysine is an inhibitor of glycine transporter 2a (GlyT2a). It selectively inhibits GlyT2a (IC50 = 48.3 nM) over GlyT1b (IC50 = >3,000 nM) in Xenopus oocytes expressing the human transporters. Oleoyl-D-lysine (30 mg/kg, i.p.) reduces allodynia in a nerve ligation rat model of neuropathic pain.