HS024 是一种选择性的 MC4 受体拮抗剂，对 MC4、MC5、MC3 和 MC1 的 Ki 分别为 0.29、3.29、5.45 和 18.6 nM。HS024 增加食物摄入。
货号:ajcx36330
CAS:N/A
分子式:C60H80F3N19O12S2
分子量：1380.52
溶解度:H2O : 50 mg/mL (36.22 mM; Need ultrasonic)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

HS024 is a selective MC4 receptor antagonist, with Kis of 0.29, 3.29, 5.45, 18.6 nM for MC4, MC5, MC3, and MC1, respectively. HS024 increase food intake[1].

[1]. Kask A, et al. Discovery of a novel superpotent and selective melanocortin-4 receptor antagonist (HS024): evaluation in vitro and in vivo. Endocrinology. 1998;139(12):5006-5014.