BZAD-01 是一种有效的，选择性和具有口服活性的 NMDA NR2B 抑制剂，Ki 值为 72 nM。BZAD-01 可以改善姿势不对称以及阿扑吗啡引起的旋转。
货号:ajcx37880
CAS:305339-41-7
分子式:C16H12F6N2O
分子量：362.27
溶解度:Methanol : 250 mg/mL (690.09 mM; Need ultrasonic)|DMSO : 100 mg/mL (276.04 mM; Need ultrasonic)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

BZAD-01 is a potent, selective and orally active inhibitor of NMDA NR2B subunit, with a Ki of 72 nM. BZAD-01 can improve postural asymmetry as well as Apomorphine-induced rotation[1].

[1]. Truong L, et, al. Behavioural effects of a selective NMDA NR1A/2B receptor antagonist in rats with unilateral 6-OHDA+parafascicular lesions. Brain Res Bull. 2009 Feb 16;78(2-3):91-6.