SETD2-IN-1 TFA 是一种有效、选择性和具有口服活性的人类组蛋白甲基转移酶 SETD2 抑制剂。SETD2-IN-1 TFA 具有抗增殖作用。
货号:ajcx33954
CAS:2411759-92-5
分子式:C24H30F4N4O4
分子量：514.51
溶解度:DMSO : 200 mg/mL (388.72 mM; Need ultrasonic)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. SETD2-IN-1 TFA has anti-proliferative effects[1].

[1]. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1.