LPA2 antagonist 2 (H2L 5226501) 是一种选择性 LPA2 拮抗剂，IC50 为 28.3 nM，比 LPA3 (IC50 为 13.85 μM) 选择性高 480 倍以上。
货号:ajcx15630
CAS:36840-10-5
分子式:C20H16N2O6
分子量：380.35
溶解度:DMSO: 83.33 mg/mL (219.09 mM)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is ＞480-fold more selective than LPA3 (IC50 of 13.85 μM)[1].

[1]. Fells JI, et al. Identification of non-lipid LPA3 antagonists by virtual screening. Bioorg Med Chem. 2008 Jun 1;16(11):6207-17.