EHMT2-IN-2是一种有效的EHMT抑制剂，对对EHMT1多肽,EHMT2多肽和细胞内EHMT2的IC50值均小于100nM。可用于血液疾病或癌症的研究。
CAS：2230850-47-0
分子式：C21H22N6O
分子量：374.44
纯度：98%
存储：Store at -20°C

Background:

EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer[1]. EHMTI PEP|<100 nM (IC50)|EHMT2 PEP|<100 nM (IC50)|EHMT2 ICW|<100 nM (IC50)

EHMT2-IN-2 (Compound 200) is a potent EHMT inhibitor, with IC50s of all< 100 nM for EEHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].

[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1.