EHMT2-IN-1是一种有效的EHMT抑制剂，对EHMT1多肽,EHMT2多肽和细胞内EHMT2的IC50均小于100nM。用于血液疾病或癌症的研究。
CAS：2230849-55-3
分子式：C18H23N7O
分子量：353.42
纯度：98%
存储：Store at -20°C

Background:

EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1]. EHMTI PEP|<100 nM (IC50)|EHMT2 PEP|<100 nM (IC50)|EHMT2 ICW|<100 nM (IC50)

EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].

[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1