生物活性
Mosapride citrate起5-HT4受体激动剂和5-HT3受体拮抗剂的作用。
靶点信息
化学数据
| 目录号 | A10607 |
| 作用机制 | Agonist (激动剂) |
| M. Wt | 614.0 |
| Formula | C21H25ClFN3O3.C6H8O7 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
| CAS No. | 112885-42-4 |
| Synonyms | TAK-370, AS-4370, Gasmotin |
| SMILES | CCOC1=CC(=C(C=C1C(=O)NCC2CN(CCO2)CC3=CC=C(C=C3)F)Cl)N.C(C(=O)O)C(CC(=O)O)(C(=O)O)O |
溶解度
| In vitro | DMSO | 77 mg/mL (125.4 mM) |
| Water | Insoluble |
| Ethanol | Insoluble |
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
储备液配制
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
| 0.1 mM | 16.29 mL | 81.43 mL | 162.87 mL |
| 0.5 mM | 3.26 mL | 16.29 mL | 32.57 mL |
| 1 mM | 1.63 mL | 8.14 mL | 16.29 mL |
| 5 mM | 0.33 mL | 1.63 mL | 3.26 mL |
*The above data is based on the productmolecular weight 614.0 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
m.cnreagent.com