CB2R-IN-1是一种有效的cannabinoidCB2受体反向激动剂，Ki为0.9nM。
CAS：1257555-79-5
分子式：C23H27F3N4O6S3
分子量：608.67
纯度：98%
存储：Store at -20°C

Background:

CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.

CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].

[1]. Tong L, et al. Expansion of SAR studies on triaryl bis sulfone cannabinoid CB2 receptor ligands. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6785-9.