Carbetocin is a novel and potent obstetric drug acting as an agonist of the oxytocin receptor (Ki of 7.1 nM) with improved in vivo stability over oxytocin. Carbetocin has high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 μM). Carbetocin has the potential for postpartum hemorrhage research. Carbetocin can crosse the blood-brain barrier and produces antidepressant-like activity via activation of oxytocin receptors in the CNS.

纯度：≥98%

CAS：37025-55-1