(E/Z)-GSK5182 is a racemic mixture of (E)-GSK5182 and (Z)-GSK5182 configurational isomers. GSK5182 is a highly specific and orally bioavailable inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma.

纯度：≥98%

CAS：1936468-29-9