Raclopride tartrate

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Raclopride tartrate

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

98185-20-7

包装与价格：

包装	价格(元)
100mg	电议
250mg	电议
500mg	电议

产品介绍

Raclopride tartrate是一种选择性的多巴胺D₂/D₃受体拮抗剂，具有抗精神作用。Raclopride tartrate 结合到D₂和D₃受体，K_i分别为 1.8 nM 和 3.5 nM。

生物活性

Raclopride tartrate is a selectivedopamine D₂/D₃receptorantagonist with potential antipsychotic effects. Raclopride tartrate binds toD₂andD₃receptors withK_is of 1.8 nM and 3.5 nM, respectively^[1]^[2].

IC₅₀& Target^[1]

D₂Receptor

1.8 nM (Ki)

D₃Receptor

3.5 nM (Ki)

D₄Receptor

2400 nM (Ki)

D₁Receptor

18000 nM (Ki)

体内研究
(In Vivo)

Raclopride tartrate (0.1, 0.3, or 0.6 mg/kg; IP; 30 min; albino male mice of the OF1 strain) significantly reduces time allocated to attack behavior^[2].

Clinical Trial

分子量

497.32

Formula

C₁₉H₂₆Cl₂N₂O₉

CAS 号

98185-20-7

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.