(R)-Phenylpiracetam (MRZ 9547) is adopamine transporter(DAT) inhibitor (K_i: 14.8 μM;IC₅₀: 65.5 μM). (R)-Phenylpiracetam can be used for the research of the neurological or neuropsychiatric disorders^[1][2].

Ki: 14.8 μM (DAT); IC50: 65.5 μM (DAT)^[2]

(R)-Phenylpiracetam displaces the binding of [¹²⁵I] RTI-55 (IC₅₀= 4.82 μM) to human recombinant DAT expressed in CHO-K1 cells^[2].

(R)-Phenylpiracetam (50 mg/kg; p.o. or i.p.; single-dose) reaches the mouse brain tissue 15 min after administration^[1].
(R)-Phenylpiracetam (10, 25, 50 mg/kg; p.o.; pretreatment for 7 days) dose-dependently reduces paw oedema and the antinociceptive response on carrageenan induced mouse^[1].

218.25

C₁₂H₁₄N₂O₂

949925-07-9

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.