CAS 862189-96-6; mirodenafil dihydrochloride

CAS:

862189-96-6

分子式:

C₂₆H₃₉Cl₂N₅O₅S

分子量:

604.59

英文名称:

mirodenafil dihydrochloride

sk 3530 dihydrochloride

sk-3530 dihydrochloride

sk3530 dihydrochloride

5-ethyl-3,5-dihydro-2-[5-[[4-(2-hydroxyethyl)-1-piperazinyl]sulfonyl]-2-propoxyphenyl]-7-propyl-4h-pyrrolo[3,2-d]pyrimidin-4-one, dihydrochloride

4-[[3-(5-ethyl-4,5-dihydro-4-oxo-7-propyl-1h-pyrrolo[3,2-d]pyrimidin-2-yl)-4-propoxyphenyl]sulfonyl]-1-piperazineethanol, dihydrochloride

5-ethyl-2-[5-[[4-(2-hydroxyethyl)piperazin-1-yl]sulfonyl]-2-propoxyphenyl]-7-propyl-3,5-dihydro-4h-pyrrolo[3,2-d]pyrimidin-4-one, dihydrochloride

用途:

Mirodenafil dihydrochloride (SK3530 dihydrochloride) 是磷酸二酯酶5（PDE-5）抑制剂，可作用于勃起功能紊乱。

推荐供应商

货号

品牌

产品名称

规格

包装、参考价格

M876958

MACKLIN

Mirodenafil dihydrochloride

≥99%

2677元/5mg; 3824元/10mg;

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储存：2-8℃

SML2955

Sigma-Aldrich

Mirodenafil dihydrochloride

≥98% (HPLC)

841.96元/10 MG; 3307.72元/50 MG;

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产品说明

生化/生理作用

Mirodenafil (SK3530) is an orally active, highly potent and selective phosphodiesterase-5 (PDE5) inhibitor (IC₅₀ = 338 pM). with therapeutic efficacy in various ED models in vivo. Comparing to sildenafil, mirodenafil shows ~10-times higher PDE5 selectivity in vitro and remains longer in the plasma and corpus cavernosum following oral dosing at 40 mg/kg in rats in vivo.

基本信息

经验(实验)分子式	C₂₆H₃₇N₅O₅S·2HCl
分子量	604.59
MDL编号	MFCD28139019

产品性质

质量水平	100
测定	≥98% (HPLC)
形式	powder
颜色	white to beige
溶解性	DMSO: 2 mg/mL, clear
储存温度	−20℃

安全信息

储存分类代码	11 - Combustible Solids
WGK	WGK 3
闪点(F)	Not applicable
闪点(C)	Not applicable