| CAS: | 19608-29-8 | |
| 分子式: | C24H34O5 | |
| 分子量: | 402.52 | |
| 英文名称: |
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| 用途: | Clascoterone (Cortexolone 17 alpha-propionate;Cortexolone 17α-propionate;CB-03-01) 是新型的局部和外周的雄性激素拮抗剂。 |
| 货号 | 品牌 | 产品名称 | 规格 | 包装、参考价格 | |||||||||||||||||||||||
| C910324 | MACKLIN | CB-03-01 | 99% | 295元/5mg; 370元/10mg; 738元/25mg; 1610元/100mg; | 咨询 | ||||||||||||||||||||||
储存:-20°C,密闭,干燥 状态:白色到米黄色粉末 | |||||||||||||||||||||||||||
| C795733 | MACKLIN | CB-03-01 | 10mM in DMSO | 198元/1ml; | 咨询 | ||||||||||||||||||||||
储存:-20°C | |||||||||||||||||||||||||||
| SML3084 | Sigma-Aldrich | Clascoterone | ≥98% (HPLC) | 780.67元/5 MG; 3157.38元/25 MG; | 咨询 | ||||||||||||||||||||||
产品说明 生化/生理作用 Clascoterone is a high-affinity androgen receptor (AR) antagonist (antiandrogen) that antagonizes testosterone-stimulated transcription activity (in reporter cells) as well as DHT-induced production of lipids and inflammatory cytokines (in human sebocytes) in cultures. When applied topically, clascoterone is as active as cyproterone acetate, and 2-, 3-, and 4-times, respectively, more active than finasteride, flutamide, and progesterone in vivo (local antiandrogenic activity in hamster′s flank organ; 100-400 μg/50 μL acetone/animal). 基本信息
产品性质
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