| CAS: | 129273-38-7 | |||||
| 分子式: | C23H31ClN4O2S | |||||
| 分子量: | 463.04 | |||||
| 英文名称: |
|
| 货号 | 品牌 | 产品名称 | 规格 | 包装、参考价格 | 详情 | ||||||||||||||||||||||||||||||||||||||||||||
| P873423 | MACKLIN | 盐酸哌罗匹隆 | 98% | 173元/200mg; 598元/1g; 2099元/5g; | 展开 | ||||||||||||||||||||||||||||||||||||||||||||
储存:2-8°C 状态:浅黄色到黄色固体 | |||||||||||||||||||||||||||||||||||||||||||||||||
| P793337 | MACKLIN | 盐酸哌罗匹隆 | 10mM in DMSO | 377元/1ml; | 展开 | ||||||||||||||||||||||||||||||||||||||||||||
储存:-20°C | |||||||||||||||||||||||||||||||||||||||||||||||||
| SML2331 | Sigma-Aldrich | Perospirone hydrochloride | ≥98% (HPLC) | 733.26元/5 MG; 2960.76元/25 MG; | 展开 | ||||||||||||||||||||||||||||||||||||||||||||
产品说明 生化/生理作用 Perospirone (SM-9018) is a typical neuroleptic (antipsychotic) agent that displays high affinity for 5-HT2, D2 and 5-HT1A receptors (Ki = 0.61, 1.4 and 2.9-1.8 nM, respectively), moderate affinity for alpha 1 and D1 receptors (Ki = 17 and 41 nM, respectively), while exhibiting much reduced affinity for alpha 2 (Ki = 408 nM) and little affinity toward muscarinic, opiate, glutamate, phencyclidine, benzodiazepine or GABAA receptors (Ki >1 μM). SM-9018 antagonizes both D2-dependent (e.g. methamphetamine-induced hyperactivity, apomorphine-induced stereotypy) and 5-HT2-mediated (e.g. tryptamine-induced clonic seizure) activities in vivo, while exhibiting very low cataleptogenic and central depressant activities commonly observed with two other neuroleptics, haloperidol and chlorpromazine. 基本信息
产品性质
安全信息
| |||||||||||||||||||||||||||||||||||||||||||||||||